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Tobacco cessation medications

Modified on Thu, Mar 9, 2023 at 3:48 PM

Drug Name

Drug Class

Indication

Route of Administration

Side Effects

Pregnancy Category

Bupropion

Atypical Antidepressant

Smoking cessation

Oral

Dry mouth, insomnia, nausea

C

Varenicline

Nicotinic Acetylcholine Receptor Partial Agonist

Smoking cessation

Oral

Nausea, insomnia, headache

C

Nicotine Gum

Nicotine Replacement Therapy

Smoking cessation

Oral

Mouth irritation, hiccups, nausea

D

Nicotine Patch

Nicotine Replacement Therapy

Smoking cessation

Transdermal

Skin irritation, insomnia, headache

D

Nicotine Lozenge

Nicotine Replacement Therapy

Smoking cessation

Oral

Mouth irritation, nausea, hiccups

D

Nicotine Inhaler

Nicotine Replacement Therapy

Smoking cessation

Inhalation

Mouth/throat irritation, cough, headache

D

Nicotine Nasal Spray

Nicotine Replacement Therapy

Smoking cessation

Nasal

Nasal irritation, cough, headache

D

Clonidine

Alpha-2 Adrenergic Agonist

Smoking cessation

Oral

Drowsiness, dry mouth, constipation

C

Nortriptyline

Tricyclic Antidepressant

Smoking cessation

Oral

Dry mouth, constipation, blurred vision

D

Gabapentin

GABA Analog

Smoking cessation

Oral

Dizziness, drowsiness, peripheral edema

C

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